Assay Detail
Binding
CHEMBL985386
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of fluorescein labeled Bax peptide from Bcl2 by fluorescence polarization assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Discovery of an orally bioavailable small molecule inhibitor of prosurvival B-cell lymphoma 2 proteins.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 19 | 8.62 | 8.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL452892 | — | — | 1 | 8.62 |
| CHEMBL444481 | — | — | 1 | - |
| CHEMBL508865 | — | — | 1 | - |
| CHEMBL448740 | — | — | 1 | - |
| CHEMBL473870 | — | — | 1 | - |
| CHEMBL451683 | — | — | 1 | - |
| CHEMBL466090 | — | — | 1 | - |
| CHEMBL469778 | — | — | 1 | - |
| CHEMBL501889 | — | — | 1 | - |
| CHEMBL376408 | ABT 737 | 1.0 | 1 | - |
| CHEMBL510761 | — | — | 1 | - |
| CHEMBL449676 | — | — | 1 | - |
| CHEMBL508864 | — | — | 1 | - |
| CHEMBL509460 | — | — | 1 | - |
| CHEMBL508093 | — | — | 1 | - |
| CHEMBL500815 | — | — | 1 | - |
| CHEMBL510351 | — | — | 1 | - |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | - |
| CHEMBL508210 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL452892 | — | Ki | = | 2.4 | nM | 8.62 |
| CHEMBL444481 | — | Ki | < | 1.0 | nM | - |
| CHEMBL508865 | — | Ki | < | 1.0 | nM | - |
| CHEMBL448740 | — | Ki | < | 1.0 | nM | - |
| CHEMBL473870 | — | Ki | < | 1.0 | nM | - |
| CHEMBL451683 | — | Ki | < | 1.0 | nM | - |
| CHEMBL466090 | — | Ki | < | 1.0 | nM | - |
| CHEMBL469778 | — | Ki | < | 1.0 | nM | - |
| CHEMBL501889 | — | Ki | < | 1.0 | nM | - |
| CHEMBL376408 | ABT 737 | Ki | < | 1.0 | nM | - |
| CHEMBL510761 | — | Ki | < | 1.0 | nM | - |
| CHEMBL449676 | — | Ki | < | 1.0 | nM | - |
| CHEMBL508864 | — | Ki | < | 1.0 | nM | - |
| CHEMBL509460 | — | Ki | < | 1.0 | nM | - |
| CHEMBL508093 | — | Ki | < | 1.0 | nM | - |
| CHEMBL500815 | — | Ki | < | 1.0 | nM | - |
| CHEMBL510351 | — | Ki | < | 1.0 | nM | - |
| CHEMBL443684 | NAVITOCLAX | Ki | < | 1.0 | nM | - |
| CHEMBL508210 | — | Ki | < | 1.0 | nM | - |