Assay Detail
Functional
CHEMBL986494
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against IRES-luciferase tagged Yellow fever virus in BHK15 cells assessed as reduction of luciferase activity after 36 hrs
39
Total Activities
39
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Yellow fever virus |
| Cell Type | BHK15 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design, synthesis, and biological evaluation of antiviral agents targeting flavivirus envelope proteins.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 39 | 4.65 | 6.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL448322 | — | — | 1 | 6.05 |
| CHEMBL476944 | — | — | 1 | 5.30 |
| CHEMBL142485 | — | — | 1 | 4.89 |
| CHEMBL518590 | — | — | 1 | 4.86 |
| CHEMBL475905 | — | — | 1 | 4.60 |
| CHEMBL517359 | — | — | 1 | 4.54 |
| CHEMBL476135 | — | — | 1 | 4.51 |
| CHEMBL503689 | — | — | 1 | 4.43 |
| CHEMBL515807 | — | — | 1 | 4.43 |
| CHEMBL478866 | — | — | 1 | 4.42 |
| CHEMBL477793 | — | — | 1 | 4.40 |
| CHEMBL375966 | — | — | 1 | 4.36 |
| CHEMBL514386 | — | — | 1 | 4.34 |
| CHEMBL477792 | — | — | 1 | 4.34 |
| CHEMBL476968 | — | — | 1 | 4.29 |
| CHEMBL478631 | — | — | 1 | - |
| CHEMBL475907 | — | — | 1 | - |
| CHEMBL475906 | — | — | 1 | - |
| CHEMBL448547 | — | — | 1 | - |
| CHEMBL478009 | — | — | 1 | - |
| CHEMBL515024 | — | — | 1 | - |
| CHEMBL478010 | — | — | 1 | - |
| CHEMBL508198 | — | — | 1 | - |
| CHEMBL513902 | — | — | 1 | - |
| CHEMBL517345 | — | — | 1 | - |
| CHEMBL515647 | — | — | 1 | - |
| CHEMBL478200 | — | — | 1 | - |
| CHEMBL479045 | — | — | 1 | - |
| CHEMBL476738 | — | — | 1 | - |
| CHEMBL517517 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL448322 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL476944 | — | EC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL142485 | — | EC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL518590 | — | EC50 | = | 13900.0 | nM | 4.86 |
| CHEMBL475905 | — | EC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL517359 | — | EC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL476135 | — | EC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL503689 | — | EC50 | = | 37000.0 | nM | 4.43 |
| CHEMBL515807 | — | EC50 | = | 37000.0 | nM | 4.43 |
| CHEMBL478866 | — | EC50 | = | 37600.0 | nM | 4.42 |
| CHEMBL477793 | — | EC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL375966 | — | EC50 | = | 44000.0 | nM | 4.36 |
| CHEMBL477792 | — | EC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL514386 | — | EC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL476968 | — | EC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL476509 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL514053 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL479029 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL478652 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL517046 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL506525 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL450900 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL505111 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL510132 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL478631 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL475907 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL475906 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL448547 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL478009 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL515024 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL478010 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL508198 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL513902 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL517345 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL515647 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL478200 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL479045 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL476738 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL517517 | — | EC50 | > | 50000.0 | nM | - |