Assay Detail
Binding
CHEMBL988089
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Binding affinity at GPR109a
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Nicotinic acid receptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.47 | 7.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL247921 | — | — | 1 | 7.14 |
| CHEMBL128604 | — | — | 1 | 6.81 |
| CHEMBL338405 | — | — | 1 | 5.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL247921 | — | Ki | = | 72.0 | nM | 7.14 |
| CHEMBL128604 | — | Ki | = | 156.0 | nM | 6.81 |
| CHEMBL338405 | — | Ki | = | 3500.0 | nM | 5.46 |