Assay Detail
Binding
CHEMBL988960
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Binding affinity to human FRK
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Assessment of chemical coverage of kinome space and its implications for kinase drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 7.57 | 8.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL450519 | — | — | 1 | 8.22 |
| CHEMBL515466 | — | — | 1 | 6.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL450519 | — | Kd | = | 6.0 | nM | 8.22 |
| CHEMBL515466 | — | Kd | = | 122.0 | nM | 6.91 |