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Assay Detail

CHEMBL991725

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of xanthine oxidase assessed as decrease of superoxide generation
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Xanthine dehydrogenase/oxidase (CHEMBL1929)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

ortho-dihydroxyisoflavone derivatives from aged Doenjang (Korean fermented soypaste) and its radical scavenging activity.
Park JS, Park HY, Kim DH, Kim DH, Kim HK.
Bioorg Med Chem Lett (2008) 18 : 5006 -5009
PubMed 18722771 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.87 5.18

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL242739 1 5.18
CHEMBL13486 1 4.78
CHEMBL1467 ALLOPURINOL 4.0 1 4.66
CHEMBL239156 1 -
CHEMBL8145 DAIDZEIN 2.0 1 -
CHEMBL513024 GLYCITEIN 1 -
CHEMBL44 GENISTEIN 2.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL242739 IC50 = 6600.0 nM 5.18
CHEMBL13486 IC50 = 16800.0 nM 4.78
CHEMBL1467 ALLOPURINOL IC50 = 21800.0 nM 4.66
CHEMBL239156 IC50 > 1000000.0 nM -
CHEMBL8145 DAIDZEIN IC50 = 429800.0 nM -
CHEMBL513024 GLYCITEIN IC50 = 682600.0 nM -
CHEMBL44 GENISTEIN IC50 = 232500.0 nM -