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Assay Detail

CHEMBL992766

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Binding
Inhibition of PARP1 in human C41 cells
41
Total Activities
41
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type C41
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Poly [ADP-ribose] polymerase 1 (CHEMBL3105)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer.
Penning TD, Zhu GD, Gandhi VB, Gong J, Thomas S, Lubisch W, Grandel R, Wernet W, Park CH, Fry EH, Liu X, Shi Y, Klinghofer V, Johnson EF, Donawho CK, Frost DJ, Bontcheva-Diaz V, Bouska JJ, Olson AM, Marsh KC, Luo Y, Rosenberg SH, Giranda VL.
Bioorg Med Chem (2008) 16 : 6965 -6975
PubMed 18541433 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 41 7.69 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL460474 1 9.00
CHEMBL453059 1 8.70
CHEMBL500298 1 8.52
CHEMBL452800 1 8.52
CHEMBL450698 1 8.40
CHEMBL452801 1 8.40
CHEMBL452025 1 8.30
CHEMBL512213 1 8.22
CHEMBL453060 1 8.22
CHEMBL460261 1 8.05
CHEMBL454180 1 8.05
CHEMBL452539 1 7.92
CHEMBL507699 1 7.92
CHEMBL508421 1 7.89
CHEMBL488664 1 7.85
CHEMBL453997 1 7.82
CHEMBL451757 1 7.82
CHEMBL452785 1 7.80
CHEMBL488831 1 7.80
CHEMBL488830 1 7.75
CHEMBL504878 1 7.75
CHEMBL513621 1 7.68
CHEMBL459853 1 7.68
CHEMBL511050 1 7.66
CHEMBL488665 1 7.62
CHEMBL488497 1 7.54
CHEMBL445724 1 7.52
CHEMBL488053 1 7.51
CHEMBL451756 1 7.12
CHEMBL81723 1 7.12

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL460474 EC50 = 1.0 nM 9.00
CHEMBL453059 EC50 = 2.0 nM 8.70
CHEMBL452800 EC50 = 3.0 nM 8.52
CHEMBL500298 EC50 = 3.0 nM 8.52
CHEMBL450698 EC50 = 4.0 nM 8.40
CHEMBL452801 EC50 = 4.0 nM 8.40
CHEMBL452025 EC50 = 5.0 nM 8.30
CHEMBL512213 EC50 = 6.0 nM 8.22
CHEMBL453060 EC50 = 6.0 nM 8.22
CHEMBL460261 EC50 = 9.0 nM 8.05
CHEMBL454180 EC50 = 9.0 nM 8.05
CHEMBL452539 EC50 = 12.0 nM 7.92
CHEMBL507699 EC50 = 12.0 nM 7.92
CHEMBL508421 EC50 = 13.0 nM 7.89
CHEMBL488664 EC50 = 14.0 nM 7.85
CHEMBL453997 EC50 = 15.0 nM 7.82
CHEMBL451757 EC50 = 15.0 nM 7.82
CHEMBL452785 EC50 = 16.0 nM 7.80
CHEMBL488831 EC50 = 16.0 nM 7.80
CHEMBL504878 EC50 = 18.0 nM 7.75
CHEMBL488830 EC50 = 18.0 nM 7.75
CHEMBL513621 EC50 = 21.0 nM 7.68
CHEMBL459853 EC50 = 21.0 nM 7.68
CHEMBL511050 EC50 = 22.0 nM 7.66
CHEMBL488665 EC50 = 24.0 nM 7.62
CHEMBL488497 EC50 = 29.0 nM 7.54
CHEMBL445724 EC50 = 30.0 nM 7.52
CHEMBL488053 EC50 = 31.0 nM 7.51
CHEMBL451756 EC50 = 76.0 nM 7.12
CHEMBL81723 EC50 = 75.0 nM 7.12
CHEMBL460060 EC50 = 94.0 nM 7.03
CHEMBL513446 EC50 = 97.0 nM 7.01
CHEMBL488496 EC50 = 160.0 nM 6.80
CHEMBL460260 EC50 = 170.0 nM 6.77
CHEMBL460267 EC50 = 180.0 nM 6.75
CHEMBL505655 EC50 = 200.0 nM 6.70
CHEMBL444135 EC50 = 210.0 nM 6.68
CHEMBL527654 EC50 = 610.0 nM 6.21
CHEMBL488052 EC50 > 1000.0 nM -
CHEMBL460259 EC50 > 1000.0 nM -
CHEMBL518484 EC50 > 1000.0 nM -