Assay Detail
Functional
CHEMBL994776
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Growth hormone secretagogue receptor type 1 (CHEMBL4616) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Aryl sulphonyl amides as potent agonists of the growth hormone secretagogue (ghrelin) receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 29 | 8.54 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL480821 | — | — | 1 | 10.30 |
| CHEMBL251572 | — | — | 1 | 9.80 |
| CHEMBL481013 | — | — | 1 | 9.80 |
| CHEMBL518774 | — | — | 1 | 9.70 |
| CHEMBL481796 | — | — | 1 | 9.60 |
| CHEMBL482220 | — | — | 1 | 9.50 |
| CHEMBL519301 | — | — | 1 | 9.40 |
| CHEMBL480037 | — | — | 1 | 9.30 |
| CHEMBL407706 | — | — | 1 | 9.10 |
| CHEMBL517543 | — | — | 1 | 9.00 |
| CHEMBL516602 | — | — | 1 | 8.90 |
| CHEMBL481620 | — | — | 1 | 8.70 |
| CHEMBL480639 | — | — | 1 | 8.60 |
| CHEMBL521246 | — | — | 1 | 8.50 |
| CHEMBL519121 | — | — | 1 | 8.40 |
| CHEMBL517391 | — | — | 1 | 8.30 |
| CHEMBL521439 | — | — | 1 | 8.20 |
| CHEMBL481408 | — | — | 1 | 8.10 |
| CHEMBL482204 | — | — | 1 | 8.10 |
| CHEMBL482203 | — | — | 1 | 8.00 |
| CHEMBL481601 | — | — | 1 | 7.80 |
| CHEMBL481014 | — | — | 1 | 7.80 |
| CHEMBL481619 | — | — | 1 | 7.70 |
| CHEMBL481602 | — | — | 1 | 7.50 |
| CHEMBL517081 | — | — | 1 | 7.50 |
| CHEMBL479865 | — | — | 1 | 6.50 |
| CHEMBL521264 | — | — | 1 | 6.40 |
| CHEMBL482194 | — | — | 1 | - |
| CHEMBL479864 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL480821 | — | EC50 | = | 0.05012 | nM | 10.30 |
| CHEMBL251572 | — | EC50 | = | 0.1585 | nM | 9.80 |
| CHEMBL481013 | — | EC50 | = | 0.1585 | nM | 9.80 |
| CHEMBL518774 | — | EC50 | = | 0.1995 | nM | 9.70 |
| CHEMBL481796 | — | EC50 | = | 0.2512 | nM | 9.60 |
| CHEMBL482220 | — | EC50 | = | 0.3162 | nM | 9.50 |
| CHEMBL519301 | — | EC50 | = | 0.3981 | nM | 9.40 |
| CHEMBL480037 | — | EC50 | = | 0.5012 | nM | 9.30 |
| CHEMBL407706 | — | EC50 | = | 0.7943 | nM | 9.10 |
| CHEMBL517543 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL516602 | — | EC50 | = | 1.259 | nM | 8.90 |
| CHEMBL481620 | — | EC50 | = | 1.995 | nM | 8.70 |
| CHEMBL480639 | — | EC50 | = | 2.512 | nM | 8.60 |
| CHEMBL521246 | — | EC50 | = | 3.162 | nM | 8.50 |
| CHEMBL519121 | — | EC50 | = | 3.981 | nM | 8.40 |
| CHEMBL517391 | — | EC50 | = | 5.012 | nM | 8.30 |
| CHEMBL521439 | — | EC50 | = | 6.31 | nM | 8.20 |
| CHEMBL481408 | — | EC50 | = | 7.943 | nM | 8.10 |
| CHEMBL482204 | — | EC50 | = | 7.943 | nM | 8.10 |
| CHEMBL482203 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL481601 | — | EC50 | = | 15.85 | nM | 7.80 |
| CHEMBL481014 | — | EC50 | = | 15.85 | nM | 7.80 |
| CHEMBL481619 | — | EC50 | = | 19.95 | nM | 7.70 |
| CHEMBL481602 | — | EC50 | = | 31.62 | nM | 7.50 |
| CHEMBL517081 | — | EC50 | = | 31.62 | nM | 7.50 |
| CHEMBL479865 | — | EC50 | = | 316.23 | nM | 6.50 |
| CHEMBL521264 | — | EC50 | = | 398.11 | nM | 6.40 |
| CHEMBL482194 | — | EC50 | > | 5011.87 | nM | - |
| CHEMBL479864 | — | EC50 | > | 5011.87 | nM | - |