Assay Detail
Binding
CHEMBL997766
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Displacement of [I125]MIT from PKR1 expressed in CHO cell membrane
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Triazine compounds as antagonists at Bv8-prokineticin receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.45 | 7.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL457515 | — | — | 1 | 7.66 |
| CHEMBL514895 | — | — | 1 | 6.36 |
| CHEMBL459142 | — | — | 1 | 5.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL457515 | — | Ki | = | 22.0 | nM | 7.66 |
| CHEMBL514895 | — | Ki | = | 440.0 | nM | 6.36 |
| CHEMBL459142 | — | Ki | = | 4719.0 | nM | 5.33 |