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Assay Detail

CHEMBL998605

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of kallikrein
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Anthranilamide-based N,N-dialkylbenzamidines as potent and orally bioavailable factor Xa inhibitors: P4 SAR.
Zhang P, Bao L, Fan J, Jia ZJ, Sinha U, Wong PW, Park G, Hutchaleelaha A, Scarborough RM, Zhu BY.
Bioorg Med Chem Lett (2009) 19 : 2186 -2189
PubMed 19297158 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.31 5.31

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL447391 1 5.31

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL447391 IC50 = 4900.0 nM 5.31