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Compound Detail

CHEMBL106109

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COC(=O)c1c(O)cccc1OCCCCNC(=O)[C@H](Cc1ccc(OCC(=O)O)cc1)NC(=O)OC(C)(C)C

Basic Information

ChEMBL ID CHEMBL106109
Phase Preclinical
Structure Type MOL
InChI Key IKOXRHVKSOJWLA-FQEVSTJZSA-N
0
Targets
4
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

560.6
MW (Da)
3.05
ALogP
9
HBA
4
HBD
169.7
PSA (Ų)
0.20
QED
1
Ro5 Violations
14
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H36N2O10
MW 560.60
Aromatic Rings 2
Heavy Atoms 40
NP-Likeness -0.41

Activity Summary

Ki 4 meas.

Literature References

PubMed DOI Target Context # Activities
- 10.1007/s00044-010-9365-7 Tyrosine-protein phosphatase non-receptor type 1 2
14592481 10.1016/j.bmcl.2003.08.064 Tyrosine-protein phosphatase non-receptor type 1 1
14592481 10.1016/j.bmcl.2003.08.064 Tyrosine-protein phosphatase non-receptor type 2 1
14592481 10.1016/j.bmcl.2003.08.064 Caco-2 1
12951078 10.1016/s0960-894x(03)00725-x Tyrosine-protein phosphatase non-receptor type 1 1
12951078 10.1016/s0960-894x(03)00725-x Tyrosine-protein phosphatase non-receptor type 22 1

Data from ChEMBL 36 via Core Engine