Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL1078126

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
C=C(C)[C@@H]1CC[C@]2(C(=O)O)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](OC(=O)Nc6ccc(-c7ccccc7)cc6)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12

Basic Information

ChEMBL ID CHEMBL1078126
Phase Preclinical
Structure Type MOL
InChI Key CHJKNYSKCNTAGY-CCSKKOMLSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

651.9
MW (Da)
11.01
ALogP
3
HBA
2
HBD
75.6
PSA (Ų)
0.32
QED
2
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C43H57NO4
MW 651.93
Aromatic Rings 2
Heavy Atoms 48
NP-Likeness 1.82

Literature References

PubMed DOI Target Context # Activities
19691293 10.1021/np900312u SW948 1
19691293 10.1021/np900312u HCT-116 1
19691293 10.1021/np900312u MDA-MB-231 1
19691293 10.1021/np900312u DNA topoisomerase 2-alpha 1
19691293 10.1021/np900312u DNA topoisomerase 1 1

Data from ChEMBL 36 via Core Engine