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Compound Detail

CHEMBL1231519

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O=c1[nH]c(=O)n([C@H]2C[C@H](O)[C@@H](COP(=O)(O)O)O2)cc1/C=C/Br

Basic Information

ChEMBL ID CHEMBL1231519
Phase Preclinical
Structure Type MOL
InChI Key LKWCVKAHHUJPQO-PIXDULNESA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

413.1
MW (Da)
-0.34
ALogP
7
HBA
4
HBD
151.1
PSA (Ų)
0.48
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C11H14BrN2O8P
MW 413.12
Aromatic Rings 1
Heavy Atoms 23
NP-Likeness 1.08

Activity Summary

IC50 1 meas. best 5.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.3 5.3 5000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 5000.0 nM 5.3 The compound was tested for inhibition of the rate of 1 uM UDP-[3H]-GlcNAc impor... 8709123

Literature References

PubMed DOI Target Context # Activities
3027328 10.1021/jm00157a022 Human alphaherpesvirus 1 3
3027328 10.1021/jm00157a022 Human alphaherpesvirus 2 3
8709123 10.1021/jm960175c Unchecked 2
3027328 10.1021/jm00157a022 Vaccinia virus 1
3027328 10.1021/jm00157a022 Vesicular stomatitis virus 1

Data from ChEMBL 36 via Core Engine