Compound Detail
CHEMBL1251
GANIRELIX 💊 Approved Drug
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💊 Approved Drug
CC/N=C(\NCC)NCCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CCCCN/C(=N/CC)NCC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@@H](Cc1cccnc1)NC(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H](Cc1ccc2ccccc2c1)NC(C)=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(N)=O
Basic Information
| ChEMBL ID | CHEMBL1251 |
| Name | GANIRELIX |
| Phase | Approved |
| Structure Type | BOTH |
| InChI Key | GJNXBNATEDXMAK-PFLSVRRQSA-N |
| Therapeutic | ✓ Yes |
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
0
Publications
2
Known Names
4
Indications
1
Mechanisms
Molecular Properties
1570.3
MW (Da)
Drug Information
| Molecule Type | Protein |
| First Approval | 1999 |
| Availability | Prescription |
| Chirality | Single Enantiomer |
Mechanism of Action
| Mechanism | Action Type | Target | Direct | Efficacy |
|---|---|---|---|---|
| Gonadotropin-releasing hormone receptor antagonist | ANTAGONIST | Gonadotropin-releasing hormone receptor | ✓ | ✓ |
Indications
Infertility, Female Reproductive Techniques, Assisted Infertility Polycystic Ovary Syndrome
ATC Classification
H01CC01
ganirelix
Level 1: SYSTEMIC HORMONAL PREPARATIONS, EXCL. SEX HORMONES AND INSULINS
Level 2: PITUITARY AND HYPOTHALAMIC HORMONES AND ANALOGUES
Data from ChEMBL 36 via Core Engine