Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL1672142

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
O=C1C(OCc2ccccc2)C(OCc2ccccc2)C[C@@H]2[C@H]3CCCN4CCC[C@@H](CN12)[C@@H]34

Basic Information

ChEMBL ID CHEMBL1672142
Phase Preclinical
Structure Type MOL
InChI Key AHHJEWZLXMNTAE-VBJCNYAASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

460.6
MW (Da)
4.26
ALogP
4
HBA
0
HBD
42.0
PSA (Ų)
0.65
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H36N2O3
MW 460.62
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness 0.87

Activity Summary

IC50 1 meas. best 5.56

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Duck hepatitis B virus
CHEMBL613761
IC50 5.56 5.56 2760.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Duck hepatitis B virus IC50 = 2760.0 nM 5.56 Antiviral activity against DHBV infected in human HepG2(2.2.15) cells assessed a... 21218816

Literature References

PubMed DOI Target Context # Activities
21218816 10.1021/jm101325h HepG2 2.2.15 1
21218816 10.1021/jm101325h Unchecked 1
21218816 10.1021/jm101325h ADMET 1
21218816 10.1021/jm101325h Duck hepatitis B virus 1

Data from ChEMBL 36 via Core Engine