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Compound Detail

CHEMBL175296

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Nc1nc(-c2ccccc2)cs1

Basic Information

ChEMBL ID CHEMBL175296
Phase Preclinical
Structure Type MOL
InChI Key PYSJLPAOBIGQPK-UHFFFAOYSA-N
0
Targets
2
Activities
1
Assay Types
0
PK Parameters
16
Publications
0
Known Names

Molecular Properties

176.2
MW (Da)
2.39
ALogP
3
HBA
1
HBD
38.9
PSA (Ų)
0.72
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C9H8N2S
MW 176.24
Aromatic Rings 2
Heavy Atoms 12
NP-Likeness -1.57

Activity Summary

IC50 2 meas.

Literature References

PubMed DOI Target Context # Activities
25559643 10.1021/jm501402x Unchecked 5
28437106 10.1021/acs.jmedchem.7b00147 Ubiquitin-conjugating enzyme E2 T 4
23526571 10.1021/ml300322n MDA-MB-231 2
- 10.6019/CHEMBL3301361 No relevant target 2
25559643 10.1021/jm501402x SPRY domain-containing SOCS box protein 2 2
10230619 10.1016/s0960-894x(99)00122-5 Unchecked 1
19419876 10.1016/j.bmc.2009.04.030 Fructose-1,6-bisphosphatase 1 1
20055453 10.1021/jm9014718 Indoleamine 2,3-dioxygenase 1 1
23000296 10.1016/j.bmc.2012.08.040 Unchecked 1
23992862 10.1016/j.bmcl.2013.07.067 L6 1
24835815 10.1016/j.ejmech.2014.04.042 Histone acetyltransferase KAT2B 1
24835815 10.1016/j.ejmech.2014.04.042 Histone acetyltransferase p300 1
25559643 10.1021/jm501402x Apical membrane antigen 1 1
25559643 10.1021/jm501402x Carbonic anhydrase 2 1
28437106 10.1021/acs.jmedchem.7b00147 Ubiquitin-conjugating enzyme E2 D3 1
28651980 10.1016/j.bmcl.2016.06.052 Indoleamine 2,3-dioxygenase 1 1

Data from ChEMBL 36 via Core Engine