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Compound Detail

CHEMBL1785001

ACETYLDIMETHYLPIPERAZINIUM IODIDE
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CC(=O)N1CC[N+](C)(C)CC1.[I-]

Basic Information

ChEMBL ID CHEMBL1785001
Name ACETYLDIMETHYLPIPERAZINIUM IODIDE
Phase Preclinical
Structure Type MOL
InChI Key VXBLRKDEHGKPAC-UHFFFAOYSA-M
Parent Compound CHEMBL356911
Active Moiety CHEMBL356911
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

157.2
MW (Da)
-0.08
ALogP
1
HBA
0
HBD
20.3
PSA (Ų)
0.45
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H17IN2O
MW 284.14
Aromatic Rings 0
Heavy Atoms 11
NP-Likeness -0.21

Activity Summary

Ki 1 meas. best 5.44

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Ki 5.44 5.44 3600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked Ki = 3600.0 nM 5.44 Displacement of [3H]epibatidine from nAChR in rat cerebral cortex 19006672

Literature References

PubMed DOI Target Context # Activities
- 10.6019/CHEMBL4495565 SARS-CoV-2 2
19006672 10.1016/j.bmc.2008.10.045 Unchecked 1
- 10.21203/rs.3.rs-23951/v1 SARS-CoV-2 1
- 10.6019/CHEMBL4495564 Replicase polyprotein 1ab 1

Data from ChEMBL 36 via Core Engine