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Compound Detail

CHEMBL1908324

METAMPICILLIN
🧪 Phase II
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🧪 Phase II
C=N[C@@H](C(=O)N[C@@H]1C(=O)N2[C@@H]1SC(C)(C)[C@@H]2C(=O)O)c1ccccc1

Basic Information

ChEMBL ID CHEMBL1908324
Name METAMPICILLIN
Phase Phase II
Structure Type MOL
InChI Key FZECHKJQHUVANE-MCYUEQNJSA-N

Known Names

Fedacilina Metampicilina Metampicillin Metampicilline Methylenampicillin Micinovo NSC-758167 Pravacilin Ruticina Viderpen
0
Targets
5
Activities
1
Assay Types
0
PK Parameters
20
Publications
10
Known Names
1
Indications

Molecular Properties

361.4
MW (Da)
1.06
ALogP
5
HBA
2
HBD
99.1
PSA (Ų)
0.60
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Chirality Racemic

Flags

Natural Product
USAN Stem -cillin

Extended Properties

Molecular Formula C17H19N3O4S
MW 361.42
Aromatic Rings 1
Heavy Atoms 25
NP-Likeness 0.65

Indications

Bacterial Infections

ATC Classification

J01CA14
metampicillin
Level 1: ANTIINFECTIVES FOR SYSTEMIC USE
Level 2: ANTIBACTERIALS FOR SYSTEMIC USE

Activity Summary

Ki 5 meas.

Literature References

PubMed DOI Target Context # Activities
37468498 10.1038/s41467-023-40064-9 Thromboxane A2 receptor 2
21741846 10.1016/j.bmc.2011.06.027 Solute carrier family 15 member 2 2
37468498 10.1038/s41467-023-40064-9 Prostaglandin G/H synthase 1 2
37468498 10.1038/s41467-023-40064-9 Alpha-1A adrenergic receptor 2
37468498 10.1038/s41467-023-40064-9 Muscarinic acetylcholine receptor M1 2
37468498 10.1038/s41467-023-40064-9 Sodium-dependent noradrenaline transporter 1
37468498 10.1038/s41467-023-40064-9 D(3) dopamine receptor 1
37468498 10.1038/s41467-023-40064-9 cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A 1
37468498 10.1038/s41467-023-40064-9 5-hydroxytryptamine receptor 1A 1
37468498 10.1038/s41467-023-40064-9 Amine oxidase [flavin-containing] A 1
37468498 10.1038/s41467-023-40064-9 Mu-type opioid receptor 1
37468498 10.1038/s41467-023-40064-9 Alpha-2A adrenergic receptor 1
37468498 10.1038/s41467-023-40064-9 Sodium-dependent serotonin transporter 1
- 10.1016/S0960-894X(97)00046-2 Adrenergic receptor beta 1
37468498 10.1038/s41467-023-40064-9 Estrogen receptor 1
37468498 10.1038/s41467-023-40064-9 Sodium-dependent dopamine transporter 1
37468498 10.1038/s41467-023-40064-9 Voltage-gated inwardly rectifying potassium channel KCNH2 1
37468498 10.1038/s41467-023-40064-9 D(1A) dopamine receptor 1
15567297 10.1016/j.ejpb.2004.07.008 Solute carrier family 15 member 2 1
15567297 10.1016/j.ejpb.2004.07.008 Solute carrier family 15 member 1 1

Data from ChEMBL 36 via Core Engine