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Compound Detail

CHEMBL1917829

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COc1ccc(-c2nc(C(=O)NN=C(C)C)cc3c2[nH]c2ccccc23)cc1

Basic Information

ChEMBL ID CHEMBL1917829
Phase Preclinical
Structure Type MOL
InChI Key WOXBIBPCPNZEOY-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
8
Publications
0
Known Names

Molecular Properties

372.4
MW (Da)
4.52
ALogP
4
HBA
2
HBD
79.4
PSA (Ų)
0.41
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H20N4O2
MW 372.43
Aromatic Rings 4
Heavy Atoms 28
NP-Likeness -0.64

Activity Summary

IC50 1 meas. best 4.39

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
UACC-62
CHEMBL614610
IC50 4.39 4.39 40710.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
UACC-62 IC50 = 40710.0 nM 4.39 Antitumor activity against human UACC62 cells by SRB colorimetric assay 21944971

Literature References

Data from ChEMBL 36 via Core Engine