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Compound Detail

CHEMBL192301

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Nc1nc(O)c2ncn(/C=C3\CC34COP(=O)(O)OC4)c2n1

Basic Information

ChEMBL ID CHEMBL192301
Phase Preclinical
Structure Type MOL
InChI Key IFLZCFZSKLISNX-QHHAFSJGSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
11
Publications
0
Known Names

Molecular Properties

325.2
MW (Da)
0.49
ALogP
9
HBA
3
HBD
145.6
PSA (Ų)
0.64
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H12N5O5P
MW 325.22
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness 0.09

Activity Summary

EC50 2 meas. best 4.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 2
CHEMBL370
EC50 4.3 4.3 50000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
15634003 10.1021/jm040149b Human alphaherpesvirus 1 3
15634003 10.1021/jm040149b Human betaherpesvirus 5 2
15634003 10.1021/jm040149b NON-PROTEIN TARGET 2
15634003 10.1021/jm040149b Human alphaherpesvirus 2 2
15634003 10.1021/jm040149b HFF 2
15634003 10.1021/jm040149b Human gammaherpesvirus 4 2
15634003 10.1021/jm040149b Hepatitis B virus 1
15634003 10.1021/jm040149b Daudi 1
15634003 10.1021/jm040149b ADMET 1
15634003 10.1021/jm040149b MEF 1
15634003 10.1021/jm040149b Molecular identity unknown 1

Data from ChEMBL 36 via Core Engine