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Compound Detail

CHEMBL19662

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CC(C)C[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NCc1cccc(Oc2ccccc2)c1)C(C)C)C(C)C)C(=O)O

Basic Information

ChEMBL ID CHEMBL19662
Phase Preclinical
Structure Type BOTH
InChI Key BZKKEMOYNVECDV-SLFDMOQUSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

904.0
MW (Da)
2.10
ALogP
11
HBA
10
HBD
304.7
PSA (Ų)
0.06
QED
3
Ro5 Violations
26
Rot. Bonds

Drug Information

Molecule Type Protein
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C46H61N7O12
MW 904.03
Aromatic Rings 3
Heavy Atoms 65
NP-Likeness -0.01

Activity Summary

IC50 2 meas. best 4.92

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.92 4.66 12000.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(00)80215-2 Unchecked 3

Data from ChEMBL 36 via Core Engine