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Compound Detail

CHEMBL1969873

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CC1(c2nc3cc(Cl)c(Cl)cc3[nH]2)CCC(CO)C(C)(C)O1

Basic Information

ChEMBL ID CHEMBL1969873
Phase Preclinical
Structure Type MOL
InChI Key MJYYHAFJMFJSDR-UHFFFAOYSA-N
3
Targets
3
Activities
1
Assay Types
0
PK Parameters
10
Publications
0
Known Names

Molecular Properties

343.2
MW (Da)
4.28
ALogP
3
HBA
2
HBD
58.1
PSA (Ų)
0.86
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H20Cl2N2O2
MW 343.25
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness 0.64

Activity Summary

EC50 3 meas. best 4.92

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Poliovirus 1
CHEMBL613556
EC50 4.92 4.92 12000.0 1
Bovine viral diarrhea virus 1
CHEMBL612571
EC50 4.34 4.34 46000.0 1
Human alphaherpesvirus 1
CHEMBL377
EC50 4.22 4.22 60000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
25082514 10.1016/j.bmc.2014.06.043 ADMET 2
25082514 10.1016/j.bmc.2014.06.043 MT4 1
25082514 10.1016/j.bmc.2014.06.043 Human immunodeficiency virus 1 1
25082514 10.1016/j.bmc.2014.06.043 Bovine viral diarrhea virus 1 1
25082514 10.1016/j.bmc.2014.06.043 NON-PROTEIN TARGET 1
25082514 10.1016/j.bmc.2014.06.043 Yellow fever virus 1
25082514 10.1016/j.bmc.2014.06.043 Reovirus sp. 1
25082514 10.1016/j.bmc.2014.06.043 Poliovirus 1 1
25082514 10.1016/j.bmc.2014.06.043 Vesicular stomatitis virus 1
25082514 10.1016/j.bmc.2014.06.043 Human alphaherpesvirus 1 1

Data from ChEMBL 36 via Core Engine