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Compound Detail

CHEMBL20579

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CC(C)C[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(=O)N1CCCC1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(C)C)C(=O)O

Basic Information

ChEMBL ID CHEMBL20579
Phase Preclinical
Structure Type MOL
InChI Key VIDIVOGMXVHHSG-AXOMYGEFSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

775.9
MW (Da)
-0.38
ALogP
10
HBA
9
HBD
286.7
PSA (Ų)
0.08
QED
2
Ro5 Violations
21
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C37H57N7O11
MW 775.90
Aromatic Rings 1
Heavy Atoms 55
NP-Likeness 0.10

Activity Summary

IC50 2 meas. best 6.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.0 5.25 1000.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(00)80215-2 Unchecked 3

Data from ChEMBL 36 via Core Engine