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Compound Detail

CHEMBL2069003

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C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@@H](CC(C)C)C(=O)OC)CC[C@@]3(C)C(CC[C@@H]4[C@@]5(C)CCC(=O)C(C)(C)C5CC[C@]43C)C12

Basic Information

ChEMBL ID CHEMBL2069003
Phase Preclinical
Structure Type MOL
InChI Key JPTHAYNSNWELKD-KFKXFZKRSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

581.9
MW (Da)
7.92
ALogP
4
HBA
1
HBD
72.5
PSA (Ų)
0.26
QED
2
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C37H59NO4
MW 581.88
Aromatic Rings 0
Heavy Atoms 42
NP-Likeness 2.30

Activity Summary

EC50 2 meas. best 4.14

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Influenza A virus
CHEMBL613740
EC50 4.14 4.14 72300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Influenza A virus EC50 = 72300.0 nM 4.14 Antiviral activity against influenza A virus determined in chicken embryo cells ... 14505668

Literature References

PubMed DOI Target Context # Activities
14505668 10.1016/s0960-894x(03)00714-5 Influenza A virus 2
14505668 10.1016/s0960-894x(03)00714-5 Human alphaherpesvirus 1 2

Data from ChEMBL 36 via Core Engine