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Compound Detail

CHEMBL2228067

6F-4Pr-D-DIBOA
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CCC(=O)ON1C(=O)COc2ccc(F)cc21

Basic Information

ChEMBL ID CHEMBL2228067
Name 6F-4Pr-D-DIBOA
Phase Preclinical
Structure Type MOL
InChI Key XUJXTRCZNMNBIH-UHFFFAOYSA-N
4
Targets
4
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

239.2
MW (Da)
1.42
ALogP
4
HBA
0
HBD
55.8
PSA (Ų)
0.78
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H10FNO4
MW 239.20
Aromatic Rings 1
Heavy Atoms 17
NP-Likeness -0.76

Activity Summary

IC50 4 meas. best 5.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Oryza sativa
CHEMBL613061
IC50 5.52 5.52 3000.0 1
Avena fatua
CHEMBL612834
IC50 5.21 5.21 6221.0 1
Echinochloa crus-galli
CHEMBL612343
IC50 5.05 5.05 9000.0 1
Triticum aestivum
CHEMBL612836
IC50 4.09 4.09 81870.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
20628996 10.1002/ps.1992 Avena fatua 4
20628996 10.1002/ps.1992 Echinochloa crus-galli 4
20628996 10.1002/ps.1992 Triticum aestivum 3
20014762 10.1021/jf903445m Lepidium sativum 2
20628996 10.1002/ps.1992 Unchecked 2
20628996 10.1002/ps.1992 Oryza sativa 2
20014762 10.1021/jf903445m Lactuca sativa 1
20014762 10.1021/jf903445m Allium cepa 1
20014762 10.1021/jf903445m Solanum lycopersicum 1

Data from ChEMBL 36 via Core Engine