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Compound Detail

CHEMBL2271644

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CCN(c1nc(Cl)nc(N[C@@H](C)c2ccccc2)n1)C(C)C

Basic Information

ChEMBL ID CHEMBL2271644
Phase Preclinical
Structure Type MOL
InChI Key XZBUOKBGYBLVFE-LBPRGKRZSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

319.8
MW (Da)
3.93
ALogP
5
HBA
1
HBD
53.9
PSA (Ų)
0.87
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H22ClN5
MW 319.84
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness -1.36

Activity Summary

IC50 2 meas. best 6.64

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Echinochloa crus-galli var. formosensis
CHEMBL2367314
IC50 6.64 6.64 229.1 1
Oryza sativa
CHEMBL613061
IC50 6.27 6.27 537.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
12400699 10.1271/bbb.66.1959 Echinochloa crus-galli var. formosensis 1
12400699 10.1271/bbb.66.1959 Oryza sativa 1

Data from ChEMBL 36 via Core Engine