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Compound Detail

CHEMBL2368272

Bruceoside-F
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CC(=O)OC(C)(C)/C(C)=C/C(=O)O[C@H]1C(=O)O[C@@H]2C[C@H]3[C@H](C)C(=O)C(O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)=C[C@]3(C)[C@H]3[C@@H](O)[C@H](O)[C@@]4(C(=O)O)OC[C@]32[C@@H]14

Basic Information

ChEMBL ID CHEMBL2368272
Name Bruceoside-F
Phase Preclinical
Structure Type MOL
InChI Key HLVUVKGKEFOUCN-RMZKDFQYSA-N
0
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

754.7
MW (Da)
-2.14
ALogP
17
HBA
7
HBD
282.3
PSA (Ų)
0.08
QED
3
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C35H46O18
MW 754.74
Aromatic Rings 0
Heavy Atoms 53
NP-Likeness 3.14

Activity Summary

EC50 1 meas.

Literature References

PubMed DOI Target Context # Activities
- 10.1016/0960-894X(96)00096-0 H9 1
- 10.1016/0960-894X(96)00096-0 Human immunodeficiency virus 1 1
- 10.1016/0960-894X(96)00096-0 ADMET 1

Data from ChEMBL 36 via Core Engine