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Compound Detail

CHEMBL2375699

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CC(=O)O[C@H]1CC[C@]2(C)[C@H]3[C@@H](O)c4c(cc(-c5cccnc5)oc4=O)O[C@]3(C)[C@@H](OC(=O)c3ccc(C#N)cc3)C[C@H]2[C@]1(C)C(=O)O

Basic Information

ChEMBL ID CHEMBL2375699
Phase Preclinical
Structure Type MOL
InChI Key JDRFTRQWGQIASU-VRKOFYPXSA-N
0
Targets
0
Activities
0
Assay Types
1
PK Parameters
2
Publications
0
Known Names

Molecular Properties

642.7
MW (Da)
4.44
ALogP
11
HBA
2
HBD
186.2
PSA (Ų)
0.37
QED
2
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C35H34N2O10
MW 642.66
Aromatic Rings 3
Heavy Atoms 47
NP-Likeness 1.40

Pharmacokinetic Data

Parameter Value Units Species
T1/2 9.0 hr Rattus norvegicus

Literature References

PubMed DOI Target Context # Activities
23535327 10.1016/j.bmcl.2013.02.088 Sterol O-acyltransferase 2 1
23535327 10.1016/j.bmcl.2013.02.088 Sterol O-acyltransferase 1 1

Data from ChEMBL 36 via Core Engine