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Compound Detail

CHEMBL2402014

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CC(C)(C)S(=O)(=O)N(CCCCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO)C1CCCCC1

Basic Information

ChEMBL ID CHEMBL2402014
Phase Preclinical
Structure Type MOL
InChI Key RWLSNJYOFAOMGC-PLACYPQZSA-N
3
Targets
3
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

464.7
MW (Da)
1.07
ALogP
7
HBA
4
HBD
121.5
PSA (Ų)
0.36
QED
0
Ro5 Violations
10
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H44N2O6S
MW 464.67
Aromatic Rings 0
Heavy Atoms 31
NP-Likeness 0.19

Activity Summary

EC50 3 meas. best 6.51

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 6.51 6.51 310.0 1
Bovine viral diarrhea virus 1
CHEMBL612571
EC50 6.51 6.51 310.0 1
Tacaribe virus
CHEMBL613131
EC50 6.4 6.4 400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
23747225 10.1016/j.bmcl.2013.04.052 ADMET 2
23747225 10.1016/j.bmcl.2013.04.052 Liver microsomes 2
23747225 10.1016/j.bmcl.2013.04.052 Tacaribe virus 1
23747225 10.1016/j.bmcl.2013.04.052 Bovine viral diarrhea virus 1 1
23747225 10.1016/j.bmcl.2013.04.052 Liver 1

Data from ChEMBL 36 via Core Engine