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Compound Detail

CHEMBL2441190

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COc1ccccc1C(=O)Nc1nc(-c2ccccn2)cs1

Basic Information

ChEMBL ID CHEMBL2441190
Phase Preclinical
Structure Type MOL
InChI Key AULRPVBCJJFDPU-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

311.4
MW (Da)
3.47
ALogP
5
HBA
1
HBD
64.1
PSA (Ų)
0.80
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H13N3O2S
MW 311.37
Aromatic Rings 3
Heavy Atoms 22
NP-Likeness -2.01

Activity Summary

EC50 1 meas. best 4.36

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vero
CHEMBL391
EC50 4.36 4.36 43500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Vero EC50 = 43500.0 nM 4.36 Cytotoxicity against african green monkey Vero cells after 72 hrs by MTT assay 24075144

Literature References

PubMed DOI Target Context # Activities
24075144 10.1016/j.bmc.2013.08.048 Mycobacterium tuberculosis 3
24075144 10.1016/j.bmc.2013.08.048 ADMET 1
24075144 10.1016/j.bmc.2013.08.048 Vero 1

Data from ChEMBL 36 via Core Engine