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Compound Detail

CHEMBL2442176

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CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC(=O)[C@H]4C[C@@H](O[Si](C)(C)C)CC[C@]4(C)[C@H]3CC[C@]12C

Basic Information

ChEMBL ID CHEMBL2442176
Phase Preclinical
Structure Type MOL
InChI Key BHEMHJCDAHJAOZ-GPVRPLDASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

474.9
MW (Da)

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C30H54O2Si
MW 474.85

Activity Summary

IC50 1 meas. best 4.42

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vero
CHEMBL391
IC50 4.42 4.42 38000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Vero IC50 = 38000.0 nM 4.42 Cytotoxicity against african green monkey Vero cells by tetrazolium dye reductio... 24084159

Literature References

PubMed DOI Target Context # Activities
24084159 10.1016/j.bmcl.2013.09.013 Unchecked 1
24084159 10.1016/j.bmcl.2013.09.013 Vero 1
24084159 10.1016/j.bmcl.2013.09.013 Mycobacterium tuberculosis 1

Data from ChEMBL 36 via Core Engine