Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL2448390

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
BOP(=O)(O)COCCn1cnc2c(N)ncnc21

Basic Information

ChEMBL ID CHEMBL2448390
Phase Preclinical
Structure Type MOL
InChI Key IGPHZMMOMQDKMT-UHFFFAOYSA-N
0
Targets
0
Activities
0
Assay Types
3
PK Parameters
17
Publications
0
Known Names

Molecular Properties

285.0
MW (Da)

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H13BN5O4P
MW 285.01

Pharmacokinetic Data

Parameter Value Units Species
T1/2 72.0 hr -
T1/2 5.3 hr -
T1/2 48.0 hr -

Literature References

PubMed DOI Target Context # Activities
17181162 10.1021/jm060030y No relevant target 8
17181162 10.1021/jm060030y ADMET 3
17181162 10.1021/jm060030y Human alphaherpesvirus 1 2
17181162 10.1021/jm060030y Sindbis virus 1
17181162 10.1021/jm060030y Hepatitis C virus 1
17181162 10.1021/jm060030y Human immunodeficiency virus 1 1
17181162 10.1021/jm060030y Vero 1
17181162 10.1021/jm060030y Punta Toro virus 1
17181162 10.1021/jm060030y Mammalian orthoreovirus 1 1
17181162 10.1021/jm060030y Human respirovirus 3 1
17181162 10.1021/jm060030y HeLa 1
17181162 10.1021/jm060030y Respiratory syncytial virus 1
17181162 10.1021/jm060030y Coxsackievirus B4 1
17181162 10.1021/jm060030y HEL 1
17181162 10.1021/jm060030y Vesicular stomatitis virus 1
17181162 10.1021/jm060030y Vaccinia virus 1
17181162 10.1021/jm060030y Human alphaherpesvirus 2 1

Data from ChEMBL 36 via Core Engine