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Compound Detail

CHEMBL3037985

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CCCCC[C@H]1C(=O)O[C@@H]2O[C@]3(C)CC[C@H]4[C@H](C)CC[C@@H]1[C@@]24OO3

Basic Information

ChEMBL ID CHEMBL3037985
Phase Preclinical
Structure Type MOL
InChI Key CBDFWIKOPAPNRI-SSGRTQLWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

338.4
MW (Da)
3.96
ALogP
5
HBA
0
HBD
54.0
PSA (Ų)
0.44
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H30O5
MW 338.44
Aromatic Rings 0
Heavy Atoms 24
NP-Likeness 3.32

Activity Summary

EC50 1 meas. best 8.05

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Plasmodium falciparum
CHEMBL364
EC50 8.05 8.05 8.9 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Plasmodium falciparum EC50 = 8.9 nM 8.05 Antimalarial activity against Plasmodium falciparum 11741486

Literature References

PubMed DOI Target Context # Activities
11741486 10.1021/jm0103007 ADMET 2
11741486 10.1021/jm0103007 Plasmodium falciparum 1
11741486 10.1021/jm0103007 BC 1
11741486 10.1021/jm0103007 Vero 1

Data from ChEMBL 36 via Core Engine