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Compound Detail

CHEMBL3105538

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COc1ccc([C@H]2O[C@@H](c3cc(OC)c(O)c(OC)c3)[C@H](C)[C@@H]2C)cc1OC

Basic Information

ChEMBL ID CHEMBL3105538
Phase Preclinical
Structure Type MOL
InChI Key AGYZMBXYRZJNNA-AHIIRKPMSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

388.5
MW (Da)
4.51
ALogP
6
HBA
1
HBD
66.4
PSA (Ų)
0.79
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C22H28O6
MW 388.46
Aromatic Rings 2
Heavy Atoms 28
NP-Likeness 0.96

Activity Summary

EC50 1 meas. best 4.94

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human gammaherpesvirus 4
CHEMBL613124
EC50 4.94 4.94 11600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Human gammaherpesvirus 4 EC50 = 11600.0 nM 4.94 Antiviral activity against EBV infected in human P3HR1 cells assessed as inhibit... 24359277

Literature References

PubMed DOI Target Context # Activities
24359277 10.1021/np400757k Unchecked 1
24359277 10.1021/np400757k ADMET 1
24359277 10.1021/np400757k Human gammaherpesvirus 4 1

Data from ChEMBL 36 via Core Engine