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Compound Detail

CHEMBL326747

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C[C@H](/N=C(\S)Nc1ccc(NC(=O)c2cscn2)nc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

Basic Information

ChEMBL ID CHEMBL326747
Phase Preclinical
Structure Type MOL
InChI Key YYLROCOWYKXSDJ-JTQLQIEISA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

519.5
MW (Da)
6.29
ALogP
5
HBA
3
HBD
79.3
PSA (Ų)
0.16
QED
2
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H15F6N5OS2
MW 519.50
Aromatic Rings 3
Heavy Atoms 34
NP-Likeness -1.69

Activity Summary

IC50 1 meas. best 8.7

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Cytomegalovirus
CHEMBL613134
IC50 8.7 8.7 2.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Cytomegalovirus IC50 = 2.0 nM 8.7 Inhibitory activity against cytomegalo virus was determined 15177441

Literature References

PubMed DOI Target Context # Activities
15177441 10.1016/j.bmcl.2004.04.093 Cytomegalovirus 1
15177441 10.1016/j.bmcl.2004.04.093 Human alphaherpesvirus 2 1
15177441 10.1016/j.bmcl.2004.04.093 Human alphaherpesvirus 3 1
15177441 10.1016/j.bmcl.2004.04.093 Respiratory syncytial virus 1
15177441 10.1016/j.bmcl.2004.04.093 Unchecked 1

Data from ChEMBL 36 via Core Engine