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Compound Detail

CHEMBL3350580

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CN1C=CCC(C(=O)OC[C@H]2O[C@@H](n3ccc(=O)[nH]c3=O)C[C@@H]2N=[N+]=[N-])=C1

Basic Information

ChEMBL ID CHEMBL3350580
Phase Preclinical
Structure Type MOL
InChI Key FQUIMJFYHVMINU-OUCADQQQSA-N
0
Targets
0
Activities
0
Assay Types
5
PK Parameters
3
Publications
0
Known Names

Molecular Properties

374.4
MW (Da)
0.78
ALogP
8
HBA
1
HBD
142.4
PSA (Ų)
0.35
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H18N6O5
MW 374.36
Aromatic Rings 1
Heavy Atoms 27
NP-Likeness 0.85

Pharmacokinetic Data

Parameter Value Units Species
AUC 4430.0 ng.hr.mL-1 -
T1/2 4.33 hr Homo sapiens
T1/2 0.56 hr Mus musculus
T1/2 0.17 hr Mus musculus
T1/2 2.13 hr -

Literature References

PubMed DOI Target Context # Activities
2374145 10.1021/jm00170a023 Mus musculus 4
2374145 10.1021/jm00170a023 ADMET 4
2374145 10.1021/jm00170a023 Homo sapiens 2

Data from ChEMBL 36 via Core Engine