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Compound Detail

CHEMBL3422487

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CN(C)CP(=O)(O)CN

Basic Information

ChEMBL ID CHEMBL3422487
Phase Preclinical
Structure Type MOL
InChI Key JUMQPEQCYCKQAL-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

152.1
MW (Da)
-0.31
ALogP
3
HBA
2
HBD
66.6
PSA (Ų)
0.54
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C4H13N2O2P
MW 152.13
Aromatic Rings 0
Heavy Atoms 9
NP-Likeness 0.17

Activity Summary

Ki 2 meas. best 5.33

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Ki 5.33 4.97 4660.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
25699141 10.1021/ml500380f Unchecked 2

Data from ChEMBL 36 via Core Engine