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Compound Detail

CHEMBL343226

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CC1CCC2C(CSCCCCCSCC3C(=O)OC4OC5(C)CCC6C(C)CCC3C46OO5)C(=O)OC3OC4(C)CCC1C32OO4

Basic Information

ChEMBL ID CHEMBL343226
Phase Preclinical
Structure Type MOL
InChI Key IYYRWMHGTXIFHA-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

696.9
MW (Da)
6.40
ALogP
12
HBA
0
HBD
108.0
PSA (Ų)
0.14
QED
3
Ro5 Violations
10
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C35H52O10S2
MW 696.93
Aromatic Rings 0
Heavy Atoms 47
NP-Likeness 1.46

Activity Summary

EC50 1 meas. best 7.92

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Plasmodium falciparum
CHEMBL364
EC50 7.92 7.92 12.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Plasmodium falciparum EC50 = 12.0 nM 7.92 Antimalarial activity against Plasmodium falciparum 11741486

Literature References

PubMed DOI Target Context # Activities
11741486 10.1021/jm0103007 Plasmodium falciparum 1

Data from ChEMBL 36 via Core Engine