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Compound Detail

CHEMBL3600899

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CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CSCC(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCN)C(N)=O)C(N)=O)C(C)C

Basic Information

ChEMBL ID CHEMBL3600899
Phase Preclinical
Structure Type MOL
InChI Key PYSXFDYFUKKAFC-XRVIBXAZSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

3110.7
MW (Da)

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C133H229N47O37S
MW 3110.65

Literature References

PubMed DOI Target Context # Activities
26094944 10.1016/j.bmc.2015.06.020 Human immunodeficiency virus 1 3
26094944 10.1016/j.bmc.2015.06.020 MT4 2
26094944 10.1016/j.bmc.2015.06.020 ADMET 1

Data from ChEMBL 36 via Core Engine