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Compound Detail

CHEMBL3686732

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CC(=O)OC1O[C@H](OC(C)=O)[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@H]1N=C=S

Basic Information

ChEMBL ID CHEMBL3686732
Phase Preclinical
Structure Type MOL
InChI Key YCFYPHXVOGTBJV-YIPFDTCYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

375.4
MW (Da)
0.13
ALogP
11
HBA
0
HBD
126.8
PSA (Ų)
0.28
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C14H17NO9S
MW 375.36
Aromatic Rings 0
Heavy Atoms 25
NP-Likeness 1.22

Activity Summary

Ki 1 meas. best 8.48

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Protein O-GlcNAcase
CHEMBL5921
Ki 8.48 8.48 3.3 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Protein O-GlcNAcase Ki = 3.3 nM 8.48 Fluorescence-Based Assay: Enzymatic reactions were carried out in a reaction con... -

Data from ChEMBL 36 via Core Engine