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Compound Detail

CHEMBL3764461

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COc1cccc(-c2nnc(/C=C/c3ccc(Br)s3)o2)c1

Basic Information

ChEMBL ID CHEMBL3764461
Phase Preclinical
Structure Type MOL
InChI Key KMWIALVZRWBPRB-SOFGYWHQSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

363.2
MW (Da)
4.74
ALogP
5
HBA
0
HBD
48.1
PSA (Ų)
0.67
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C15H11BrN2O2S
MW 363.24
Aromatic Rings 3
Heavy Atoms 21
NP-Likeness -1.60

Activity Summary

IC50 1 meas. best 4.96

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.96 4.96 11100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 11100.0 nM 4.96 Inhibition of Dengue virus 2 RdRp using homopolymeric uridine RNA as template as... 26774922

Literature References

PubMed DOI Target Context # Activities
26774922 10.1016/j.ejmech.2015.12.046 dengue virus type 2 2
26774922 10.1016/j.ejmech.2015.12.046 dengue virus type 4 2
26774922 10.1016/j.ejmech.2015.12.046 ADMET 1
26774922 10.1016/j.ejmech.2015.12.046 Unchecked 1
26774922 10.1016/j.ejmech.2015.12.046 dengue virus type 1 1
26774922 10.1016/j.ejmech.2015.12.046 dengue virus type 3 1

Data from ChEMBL 36 via Core Engine