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Compound Detail

CHEMBL3911921

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C[C@@]1(C#N)[C@@H](c2cnc3c(N)ncnn23)O[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H]1O

Basic Information

ChEMBL ID CHEMBL3911921
Phase Preclinical
Structure Type MOL
InChI Key MPTMBPALHBJNEO-UOKLYIGXSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

530.2
MW (Da)
-0.62
ALogP
14
HBA
6
HBD
282.2
PSA (Ų)
0.23
QED
3
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C12H17N6O12P3
MW 530.22
Aromatic Rings 2
Heavy Atoms 33
NP-Likeness 0.77

Activity Summary

IC50 1 meas. best 7.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Genome polyprotein
CHEMBL6040
IC50 7.3 7.3 50.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Genome polyprotein IC50 = 50.0 nM 7.3 Inhibition Assay: To measure inhibition of the enzymatic activity of the HCV NS5... -

Data from ChEMBL 36 via Core Engine