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Compound Detail

CHEMBL3941082

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Cc1cc([C@@](C)(O)C#Cc2ccc3c(c2)-c2nc(C(N)=O)c(C4CC4)n2CCO3)no1

Basic Information

ChEMBL ID CHEMBL3941082
Phase Preclinical
Structure Type MOL
InChI Key YWHACELMMCHPDB-QHCPKHFHSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
10
Publications
0
Known Names

Molecular Properties

418.4
MW (Da)
2.47
ALogP
7
HBA
2
HBD
116.4
PSA (Ų)
0.63
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H22N4O4
MW 418.45
Aromatic Rings 3
Heavy Atoms 31
NP-Likeness -1.00

Literature References

PubMed DOI Target Context # Activities
31531194 10.1021/acsmedchemlett.8b00658 ADMET 3
31531194 10.1021/acsmedchemlett.8b00658 Serine/threonine-protein kinase D1 2
31531194 10.1021/acsmedchemlett.8b00658 No relevant target 2
31531194 10.1021/acsmedchemlett.8b00658 Mitogen-activated protein kinase kinase kinase 14 1
31531194 10.1021/acsmedchemlett.8b00658 Unchecked 1
31531194 10.1021/acsmedchemlett.8b00658 RAC-alpha serine/threonine-protein kinase 1
31531194 10.1021/acsmedchemlett.8b00658 Tyrosine-protein kinase JAK1 1
31531194 10.1021/acsmedchemlett.8b00658 Mitogen-activated protein kinase kinase kinase kinase 4 1
31531194 10.1021/acsmedchemlett.8b00658 Misshapen-like kinase 1 1
31531194 10.1021/acsmedchemlett.8b00658 Serine/threonine-protein kinase PAK 4 1

Data from ChEMBL 36 via Core Engine