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Compound Detail

CHEMBL4083048

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CC[C@H](C)[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@@H]2CSSC[C@H](NC1=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(=O)O)C(=O)NCC(=O)N[C@@H](CCCNC(=N)N)C(=O)N2

Basic Information

ChEMBL ID CHEMBL4083048
Phase Preclinical
Structure Type MOL
InChI Key SJOQDGYJJVWVGL-MRZDYPPISA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

1715.0
MW (Da)

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C79H107N23O17S2
MW 1715.00

Literature References

PubMed DOI Target Context # Activities
29605997 10.1021/acs.jmedchem.8b00170 Melanocortin receptor 4 4
29605997 10.1021/acs.jmedchem.8b00170 Melanocortin receptor 3 3
29605997 10.1021/acs.jmedchem.8b00170 Melanocyte-stimulating hormone receptor 3
29605997 10.1021/acs.jmedchem.8b00170 Melanocortin receptor 5 2
29605997 10.1021/acs.jmedchem.8b00170 No relevant target 1

Data from ChEMBL 36 via Core Engine