Compound Detail
CHEMBL408877
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Basic Information
| ChEMBL ID | CHEMBL408877 |
| Phase | Preclinical |
| Structure Type | BOTH |
| InChI Key | GDEKXRXZCJGVLW-IZIWSLEDSA-N |
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names
Molecular Properties
1869.2
MW (Da)
Drug Information
| Molecule Type | Protein |
| Availability | Unknown |
| Chirality | Unknown |
Activity Summary
Kd 1 meas. best 7.6
Target Activity Profile
| Target | Type | Best pChEMBL | Mean pChEMBL | Best (nM) | # Data |
|---|---|---|---|---|---|
| Protein Tat CHEMBL4609 | Kd | 7.6 | 7.6 | 25.0 | 1 |
Activity Data Samples
Top measurements by pChEMBL value
| Target | Type | Rel. | Value | Units | pChEMBL | Assay | PubMed |
|---|---|---|---|---|---|---|---|
| Protein Tat | Kd | = | 25.0 | nM | 7.6 | Dissociation constant for TAR RNA | 11229778 |
Literature References
| PubMed | DOI | Target Context | # Activities |
|---|---|---|---|
| 11229778 | 10.1016/s0960-894x(01)00005-1 | Protein Tat | 1 |
Data from ChEMBL 36 via Core Engine