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Compound Detail

CHEMBL4115685

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CC1=CCC(CC(C)Oc2ccc(/C=C3\SC(O)=NC3=O)cc2)CC1

Basic Information

ChEMBL ID CHEMBL4115685
Phase Preclinical
Structure Type MOL
InChI Key KCXMCDKKIBWBCH-PDGQHHTCSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

357.5
MW (Da)
5.12
ALogP
3
HBA
1
HBD
58.9
PSA (Ų)
0.59
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H23NO3S
MW 357.48
Aromatic Rings 1
Heavy Atoms 25
NP-Likeness -0.01

Activity Summary

IC50 1 meas. best 7.55

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
CHEMBL1293255
IC50 7.55 7.55 28.4 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine