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Compound Detail

CHEMBL4115690

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O=C1N=C(O)S/C1=C\c1cccc(OCCCCC2CCCCC2)c1Cl

Basic Information

ChEMBL ID CHEMBL4115690
Phase Preclinical
Structure Type MOL
InChI Key NLKDKIPMGJWXBJ-LGMDPLHJSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

393.9
MW (Da)
6.00
ALogP
3
HBA
1
HBD
58.9
PSA (Ų)
0.46
QED
1
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H24ClNO3S
MW 393.94
Aromatic Rings 1
Heavy Atoms 26
NP-Likeness -0.61

Activity Summary

IC50 1 meas. best 7.03

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
CHEMBL1293255
IC50 7.03 7.03 94.5 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine