Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL413393

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
COc1ccc(C(=O)CC[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CO)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@H](Cc2ccc(Cl)cc2)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(C)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N2CCC[C@@H]2C(=O)N[C@@H](C)C(N)=O)cc1

Basic Information

ChEMBL ID CHEMBL413393
Phase Preclinical
Structure Type BOTH
InChI Key UFOMLGCSEHLELA-NQZTYIJCSA-N
0
Targets
2
Activities
2
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

1486.1
MW (Da)

Drug Information

Molecule Type Protein
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C73H97ClN18O14
MW 1486.14

Activity Summary

Kd 1 meas.
Ki 1 meas.

Literature References

PubMed DOI Target Context # Activities
7510341 10.1021/jm00031a021 Rattus norvegicus 2
7510341 10.1021/jm00031a021 Gonadotropin-releasing hormone receptor 1

Data from ChEMBL 36 via Core Engine