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Compound Detail

CHEMBL4205122

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COc1ccc(/C=C/C(=O)O[C@H]2[C@@H]3C=CO[C@@H](O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)[C@@H]3[C@@]3(CO)O[C@@H]23)cc1

Basic Information

ChEMBL ID CHEMBL4205122
Phase Preclinical
Structure Type MOL
InChI Key SYHPDMZDZYFZLU-WEWXOPRLSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

522.5
MW (Da)
-1.32
ALogP
12
HBA
5
HBD
176.9
PSA (Ų)
0.15
QED
2
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C25H30O12
MW 522.50
Aromatic Rings 1
Heavy Atoms 37
NP-Likeness 2.54

Activity Summary

IC50 1 meas. best 4.11

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
IC50 4.11 4.11 78500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
No relevant target IC50 = 78500.0 nM 4.11 Peroxynitrite scavenging activity assessed as inhibition of DHR 123 oxidation af... 28787158

Literature References

PubMed DOI Target Context # Activities
28787158 10.1021/acs.jnatprod.7b00139 No relevant target 1

Data from ChEMBL 36 via Core Engine