Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL4205659

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
COc1c2c(c(O)c3c1[C@H](O)Cc1cc(CC(C)=O)c(C(=O)O)c(O)c1-3)C(=O)c1cccc(O)c1C2=O

Basic Information

ChEMBL ID CHEMBL4205659
Phase Preclinical
Structure Type MOL
InChI Key IKBVYLJFSULGQO-CQSZACIVSA-N
1
Targets
3
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

504.4
MW (Da)
2.67
ALogP
9
HBA
5
HBD
178.7
PSA (Ų)
0.28
QED
1
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C27H20O10
MW 504.45
Aromatic Rings 3
Heavy Atoms 37
NP-Likeness 1.73

Activity Summary

EC50 3 meas. best 4.6

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
EC50 4.6 4.6 25000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
No relevant target EC50 = 25000.0 nM 4.6 Antioxidant activity assessed as DPPH radical scavenging activity incubated for ... 30178674

Literature References

PubMed DOI Target Context # Activities
30178674 10.1021/acs.jnatprod.8b00397 No relevant target 3

Data from ChEMBL 36 via Core Engine