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Compound Detail

CHEMBL4227619

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CN1CCN(C(=O)C[C@H](NC(=O)c2ccc(-c3ccccc3)cc2)C(=O)NC2(C#N)CC2)CC1

Basic Information

ChEMBL ID CHEMBL4227619
Phase Preclinical
Structure Type MOL
InChI Key OADOPEZAMOOIHQ-QFIPXVFZSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

459.6
MW (Da)
1.79
ALogP
5
HBA
2
HBD
105.5
PSA (Ų)
0.66
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C26H29N5O3
MW 459.55
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness -0.95

Literature References

PubMed DOI Target Context # Activities
29615344 10.1016/j.bmcl.2018.03.069 Cathepsin S 1
29615344 10.1016/j.bmcl.2018.03.069 Procathepsin L 1
29615344 10.1016/j.bmcl.2018.03.069 Cathepsin K 1
29615344 10.1016/j.bmcl.2018.03.069 Cathepsin B 1
29615344 10.1016/j.bmcl.2018.03.069 Falcipain 2 1

Data from ChEMBL 36 via Core Engine